3
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T13425 | (1S,3R,5R)-PIM447 dihydrochloride | (1S,3R,5R)-LGH447 dihydrochloride | CDK |
(1S,3R,5R)-PIM447 (dihydrochloride) an inhibitor of PIM(IC50 of 0.095 μM for Pim1, 0.522 μM for Pim2 and 0.369 μM for Pim3). | |||
T12473 | PIM-447 dihydrochloride | LGH447 dihydrochloride | Others |
PIM-447 dihydrochloride is an orally available and selective inhibitor of pan-PIM kinase(Ki values of 6, 18, and 9 pM for PIM1, PIM2, and PIM3, respectively). | |||
T63550 | (1S,3R,5R)-PIM447 dihydrochloride | ||
(1S,3R,5R)-PIM447 (dihydrochloride) is an inhibitor of PIM, capable of Pim1 (IC50: 0.095 μM), Pim2 (IC50: 0.522 μM) and Pim3 (IC50: 0.369 μM). |